In Vitro ADME, CYP & Metabolism Assays Vendors

Compare labs for in vitro ADME and metabolism assays: metabolic stability, protein binding, permeability, CYP inhibition and induction, metabolite profiling.

Related workflows

Inotiv is a CRO and research models provider offering toxicology, in vivo pharmacology, research and transgenic models, bioanalysis and DMPK.

Products: Teklad, Target Sufficiency +1 more

Evidence-backed capability match
Matches In Vitro ADME, CYP & Metabolism Assays
“Accelerate your drug development with Inotiv's tailored in vitro DMPK package. Our team of experienced scientists leverages state-of-the-art facilities and proven methodologies to…”
Source: inotiv.com

Also offers: Toxicology Studies, In Vivo Pharmacology & Efficacy Models, +3 more

Frontage Laboratories is a CRO and CDMO providing bioanalysis, DMPK and ADME studies, toxicology, Phase I support, and drug manufacturing.
Evidence-backed capability match
Matches In Vitro ADME, CYP & Metabolism Assays
“Frontage Global Drug Discovery Services (GDDS) offers a full spectrum of in vitro ADMET assays, including metabolic stability, drug-drug internation with P450 and transporters…”
Source: frontagelab.com

Also offers: Bioanalysis & Biomarker Assay Services, Integrated CDMO/CMO Services, +3 more

Crown Bioscience is a translational oncology CRO offering in vivo efficacy studies, PDX and cancer models, biomarker discovery, and clinical biomarker testing.

Products: OrganoidXplore, HuGEMM +3 more

Evidence-backed capability match
Matches In Vitro ADME, CYP & Metabolism Assays
“Metabolic stability (Liver microsomes, S9, hepatocytes)”
Source: crownbio.com

Also offers: In Vivo Pharmacology & Efficacy Models, Oncology Models & PDX Studies, +2 more

Altasciences is an early phase CRO and CDMO providing toxicology, IND-enabling studies, clinical pharmacology, bioanalysis, and drug manufacturing.

Products: Acceleration Platform

Evidence-backed capability match
Matches In Vitro ADME, CYP & Metabolism Assays
“In vitro plasma stability, metabolite identification, and plasma protein binding studies using mass spectrometry platforms”
Source: altasciences.com

Also offers: Toxicology Studies, First-in-Human (Phase I) Clinical Pharmacology Support, +2 more

BioIVT supplies human and animal biospecimens, hepatocytes, PBMCs and other primary cells, plus ADME, DDI, bioanalysis and in vitro assay services.
Evidence-backed capability match
Matches In Vitro ADME, CYP & Metabolism Assays
“…| | In vitro ADME studies such as evaluation of metabolic stability, metabolite profiling, CYP enzyme inhibition and induction | | | Assessing (long term) off-target effects…”
Source: bioivt.com

Also offers: Cell Culture, Cell Models & Organoid Products, Human Biospecimens & Biobank Samples, +2 more

Celerion is a CRO and laboratory services provider supporting clinical development, bioanalysis, biometrics, trial operations, and regulatory submissions.

Products: ClinQuick

Evidence-backed capability match
Matches In Vitro ADME, CYP & Metabolism Assays
“In vitro cross-species metabolism and metabolite identification using hepatocytes, liver microsomes, and S9 fractions”
Source: celerion.com

Also offers: First-in-Human (Phase I) Clinical Pharmacology Support, Clinical Trial Bioanalytical & Biomarker Testing, +2 more

Compare listed vendors

What this covers: In vitro ADME and metabolism assays such as microsomal stability, hepatocyte stability, plasma protein binding, permeability, CYP inhibition/induction, and metabolite profiling.

VendorDelivery modelAlso offersIn their words
AltasciencesCRO / Research Services ProviderDrug Metabolism, Pharmacokinetics & ADME Studies, Pharmacokinetics & PK/PD Modeling“In vitro plasma stability, metabolite identification, and plasma protein binding studies using mass spectrometry platforms”altasciences.com · reviewed Oct 21, 2026
BioIVTProduct / Instrument SupplierDrug Metabolism, Pharmacokinetics & ADME Studies, Drug-Drug Interaction & Transporter Studies“…| | In vitro ADME studies such as evaluation of metabolic stability, metabolite profiling, CYP enzyme inhibition and induction | | | Assessing (long term)…”bioivt.com · reviewed Oct 25, 2026
CelerionCRO / Research Services Provider—“From early in vitro metabolism through non-clinical ADME and human pharmacology studies, we establish a connection between what is formed in vitro, what is…”celerion.com · reviewed Oct 28, 2026
Crown BioscienceCRO / Research Services ProviderDrug Metabolism, Pharmacokinetics & ADME Studies, Pharmacokinetics & PK/PD Modeling“Metabolic stability (Liver microsomes, S9, hepatocytes)”crownbio.com · reviewed Oct 21, 2026
Frontage LaboratoriesCRO / Research Services ProviderDrug Metabolism, Pharmacokinetics & ADME Studies, Drug-Drug Interaction & Transporter Studies, Pharmacokinetics & PK/PD Modeling“Frontage Global Drug Discovery Services (GDDS) offers a full spectrum of in vitro ADMET assays, including metabolic stability, drug-drug internation with P450…”frontagelab.com · reviewed Oct 21, 2026
InotivCRO / Research Services ProviderDrug Metabolism, Pharmacokinetics & ADME Studies, Drug-Drug Interaction & Transporter Studies, Pharmacokinetics & PK/PD Modeling“Accelerate your drug development with Inotiv's tailored in vitro DMPK package. Our team of experienced scientists leverages state-of-the-art facilities and…”inotiv.com · reviewed Oct 21, 2026